Picamilon Sodium (Nicotinoyl-GABA)
AUD25
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Picamilon is a synthetic molecular conjugate. It contains Y-aminobutyric acid (GABA) and niacin (vitamin B3). This chemical design is intended to alter pharmacokinetic properties relative to individual components. Picamilon is studied in mechanistic research contexts to explore how chemical linkage influences:
- compound distribution
- receptor interactions
- and molecular signaling pathways.
The compound has been used as a reference material in laboratory settings to probe neuronal receptor interactions and transporter dynamics.
Chemical and Molecular Properties
| Property | Description |
| Compound Name | N-nicotinoyl-Y-aminobutyric acid (Picamilon) |
| Synonyms | Nicotinoyl-GABA; Pikamilon; Pikatropin |
| Molecular Formula | C10H12N2O3 |
| Molecular Weight | ~208.21 g/mol |
| CAS Number | 34562-97-5 |
| Structural Class | GABA derivative/niacin conjugate |
| Chemical Nature | Synthetic small molecule |
| Research Classification | Neuronal signaling and transport investigational compound |
Working Mechanism of Picamilon
Molecular Conjugation and Transport
Picamilon is structurally composed of the inhibitory neurotransmitter analogue Y-aminobutyric acid (GABA) chemically linked to niacin. This design alters lipophilicity relative to GABA alone. It has been investigated in preclinical research for its ability to influence membrane permeability in controlled experimental systems.
Interaction with GABA-Related Targets
GABA itself exhibits specific interactions with GABA receptor subtypes. Recent assays also indicate that Picamilon, despite structural similarity, does not exhibit high affinity across a panel of 50 biological targets, including major ion channels, transporters, and receptor proteins at typical in vitro screening concentrations. This suggests that the mechanisms of action in mechanistic studies may involve indirect modulation or metabolic transformation in experimental preparations rather than direct receptor agonism.
Metabolic Transformation in Experimental Models
In controlled research environments, Picamilon has been observed to be hydrolyzed into its constituent moieties – GABA and niacin – under specific conditions. These component molecules can then be evaluated independently for receptor interaction profiles and signaling effects in mechanistic assays.
Picamilon Research Applications (Laboratory Use Only)
- In vitro studies of inhibitor and transporter activity related to GABA analogues
- Experimental evaluation of compound distribution and membrane permeability
- Biochemical assays of metabolic breakdown products (GABA and niacin)
- Mechanistic receptor binding profiling using high-throughput screening methods
These applications are strictly confined to laboratory research and analytical investigations.
Why Choose Purerawz for Picamilon?
Buy Picamilon (N-nicotinoyl-Y-aminobutyric acid) for laboratory research use from our online shop. At Purerawz, we provide high-quality reference materials. Each research compound comes with a Certificate of Analysis for verification of purity and concentration.
Note: Picamilon is an investigational compound currently undergoing scientific evaluation and has not been established as safe or effective for any therapeutic use.
Disclaimer
This information is for educational purposes only and not medical advice. Products are for research use only. Research must follow IRB or IACUC guidelines. Verify information independently before purchasing. By ordering, you agree to our Terms and Conditions.
ATTENTION: All our products are for LABORATORY AND RESEARCH PURPOSES ONLY, not for veterinary or human use.
Frequently Asked Questions
What is Picamilon Sodium (Nicotinoyl-GABA)?
Picamilon Sodium is a conjugate of niacin and GABA (nicotinoyl-GABA), studied for its combined structural properties in research settings. It is supplied strictly as a laboratory research reference material and is not intended for human or veterinary use.
Can Picamilon Sodium (Nicotinoyl-GABA) be imported or is it legal in Australia?
This compound is offered solely for laboratory research use and is not for human consumption. Research chemicals of this type may be subject to import and supply restrictions, so researchers must confirm the current regulatory and import status in their jurisdiction before ordering.
How is Picamilon Sodium (Nicotinoyl-GABA) tested?
Identity and purity are established through independent third-party analysis using HPLC and mass spectrometry. A batch-specific certificate of analysis (COA) documenting a purity of at least 99% is supplied.
How should Picamilon Sodium (Nicotinoyl-GABA) be stored in the laboratory?
It is typically stored as a dry powder in a sealed container kept cool and away from light and moisture to maintain stability. Storage conditions should follow the parameters recorded on the accompanying certificate of analysis.
For laboratory and research use only. This product is not for human or veterinary consumption, and nothing on this page is medical advice. Researchers are responsible for compliance with all applicable Australian laws (including TGA regulations) and institutional guidelines.
| Form | Powder |
|---|---|
| Strength | 5g |
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